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Table 1 In vitro drug response of MLH1−/− cell lines

From: Chemo-immunotherapy improves long-term survival in a preclinical model of MMR-D-related cancer

Drug

IC50 value [μM]

MLH1−/− A7450 T1 M1a

MLH1−/−  328

MLH1−/−  1351

GEM

0.05

0.07

< 0.02

Cisplatin

0.63

0.05

0.06

5-FU

2.15

3.57

1.00

CPX

> 300

> 300

> 300

  1. GEM Gemcitabin, 5-FU 5-Fluorouracil, CPX Cyclophosphamide; a [18]